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目录号 | 产品名称 | 产品描述 |
R21122038 | NPY5RA972 | NPY5RA972 is a neuropeptide Y Y5 antagonist. |
R21122039 | ASP 2905 | ASP2905 是由 Kcnh3/BEC1 基因编码的有效且选择性的钾通道 Kv12.2 抑制剂。ASP2905 可以穿越血脑屏障并具有抗精神病活性。 |
R21122040 | CID 2745687 | CID 2745687 is a GPR35 antagonist that inhibited the effects at human GPR35 of c |
R21122041 | KPT251 | KPT-251 is a selective nuclear export inhibitor. |
R21122042 | LEI110 | LEI110(LEI-110)是一种有效的磷脂酶A2组XVI(PLA2G16)抑制剂,Ki为20 nM,对HRASLS2,RARRES3和iNAT也有活性(pI |
R21122043 | MYLS22 | MYLS22 是首创的,选择性视神经萎缩 1 (OPA1) 抑制剂。MYLS22 可以靶向内皮细胞 OPA1 减少肿瘤的生长,通过影响 NFkB 活性和血管生成 |
R21122044 | APX001 | APX001(APX 001A;E1210)是一种新型广谱抗真菌剂,可抑制真菌蛋白Gwt1,显示出显着的活性MIC50和MIC90值0.004和0.031 ug |
R21122045 | DoPAT | |
R21122046 | (S)FTY720 Phosphate | FTY720 (S)-Phosphate 是一种 S1P 受体 1 (S1PR1) 激动剂,可以用于急性肺损伤等急性炎症的研究。 |
R21122047 | CYM50769 (ML250) | neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist |
R21122048 | CAY10526 | CAY10526 is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB |
R21122049 | NSC-13755 | |
R21122050 | ML261 | |
R21122051 | Galloflavin | Galloflavin inhibits both the A and B isoforms of lactate dehydrogenase with Ki |
R21122052 | RO2959 Hydrochloride | |
R21122053 | HA-155(Z) | HA-155 是一种高效、选择性的 ATX 抑制剂,其 IC50 值为 5.7 nM。 |
R21122054 | GSK205 | GSK205 是一种高效的,选择性的 TRPV4 拮抗剂,IC50 值为 4.19 μM,可抑制 TRPV4 介导的 Ca2+ 内流。 |
R21122055 | SOMG-833 | 一种有效的,选择性的ATP竞争性c-MET抑制剂,IC50为0.93 nM;对20种激酶组的选择性显示>10,000倍,包括c-MET家族成员RON和高度 |
R21122056 | GF-61 | |
R21122057 | LDN-211904 Oxalate | LDN-211904 is an inhibitor of erythropoietin-producing hepatocellular carcinoma |
R21122058 | ML00253764 hydrochloride | ML00253764 is a non-peptide, brain penetrant melanocortin MC4 receptor (MC4R) an |
R21122059 | NBI-35965 Mesylate | NBI-35965 Mesylate is a potent and selective corticotropin-releasing factor rece |
R21122060 | PAOPA | dopamine D2 receptor modulator. |
R21122061 | ML-211 | ML-211 is a carbamate-based dual inhibitor of LYPLA1 (IC50 = 17 nM) and the rela |
R21122062 | NSC-658497 | NSC-658497 是一种有效的 SOS1 抑制剂。NSC-658497 与 SOS1 结合,竞争性抑制 SOS1-Ras 相互作用,并呈剂量依赖性抑制 SO |