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首页 > 产品展示 > Protein Tyrosine Kinase
目录号 产品名称 产品描述
R10003 Infigratinib (Synonyms: BGJ-398; NVP-BGJ398) Infigratinib (BGJ-398; NVP-BGJ398) 是 FGFR 家族的有效抑制剂,抑制 FGFR1,FGFR2,FGFR3 和 FGFR4
R10006 Allitinib tosylate (Synonyms: AST-1306 (TsOH))/897383-62-9 游离态 Allitinib tosylate (AST-1306 TsOH) 是不可逆的EGFR和ErbB2抑制剂,IC50分别为0.5 nM和3 nM,对突变型EGF
R10036 XL880; Foretinib; GSK136308 Foretinib (GSK1363089) is an ATP-competitive inhibitor of HGFR and VEGFR, mostly
R10037 ANA12 ANA-12 is a selective TrkB antagonist with Kd of 10 nM and 12 μM for the high an
R10042 CO1686; Rociletinib Rociletinib (CO-1686, AVL-301) is an irreversible, mutant-selective EGFR inhibit
R10052 GNF-5837 GNF-5837 is a selective, and orally bioavailable pan-TRK inhibitor for TrkA, and
R10054 TAE684 TAE684 (NVP-TAE684) is a potent and selective ALK inhibitor with IC50 of 3 nM in
R10058 Masitinib Masitinib is a novel inhibitor for Kit and PDGFRα/β with IC50 of 200 nM and 540
R10061 Nexavar; Bay 43-9006; Sorafenib Sorafenib Tosylate is a multikinase inhibitor of Raf-1, B-Raf and VEGFR-2 with I
R10062 SAR131675 SAR131675是一种VEGFR3抑制剂,无细胞试验中IC50/Ki为23 nM/12 nM,作用于VEGFR3比作用于VEGFR1/2选择性高50和10倍,
R10064 Brivanib; BMS540215 Brivanib is an ATP-competitive inhibitor against VEGFR2 with IC50 of 25 nM, mode
R10076 Crizotinib; PF02341066 Crizotinib (PF-02341066) is a potent inhibitor of c-Met and ALK with IC50 of 11
R10077 AMG208 AMG 208 is a highly selective c-Met inhibitor with IC50 of 9 nM. Phase 1.
R10078 EMD1214063 Tepotinib (EMD 1214063) is a potent and selective c-Met inhibitor with IC50 of 4
R10087 AZD9291 Osimertinib (AZD9291) is an oral, irreversible, and mutant-selective EGFR inhibi
R10103 Cedirannib; AZD2171 Cediranib (AZD2171) is a highly potent VEGFR(KDR) inhibitor with IC50 of 1000-fo
R10114 PHA665752 PHA-665752 is a potent, selective and ATP-competitive c-Met inhibitor with IC50
R10115 SU11274 U11274 is a selective Met inhibitor with IC50 of 10 nM in cell-free assays, no e
R10116 OSI906 OSI-906 (Linsitinib) is a selective inhibitor of IGF-1R with IC50 of 35 nM in ce
R10118 Regorafenib; BAY73-4506; BAY734506 Regorafenib (BAY 73-4506) 是一种多靶点受体酪氨酸激酶抑制剂,抑制VEGFR1/2/3,PDGFRβ,Kit,RET 和 Raf-1 的
R10126 WZ4002 WZ4002 is a novel, mutant-selective EGFR inhibitor for EGFR(L858R)/(T790M) with
R10127 Linifanib (Synonyms: ABT-869; AL-39324) Linifanib (ABT-869) 是一种高效、口服的 VEGFR 和 PDGFR 家族多靶点抑制剂,对 KDR、FLT1、PDGFRβ、FLT3 的 IC
R10134 BMS599626 Free base AC480 (BMS-599626) is a selective and efficacious inhibitor of HER1 and HER2 wit
R10138 AV-951; Tivozanib Tivozanib (AV-951) is a potent and selective VEGFR inhibitor for VEGFR1/2/3 with
R10143 BMS907351; XL184; Cabozantinib Cabozantinib (XL184, BMS-907351) is a potent VEGFR2 inhibitor with IC50 of 0.035
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