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首页 > 产品展示 > PI3K/Akt/mTOR
目录号 产品名称 产品描述
R10009 AZD8055 AZD-8055 是一种ATP竞争性的 mTOR 抑制剂,IC50 为 0.8 nM。AZD-8055 抑制 mTORC1 和 mTORC2。 
R10011 BIO-acetoxime; GSK3 Inhibitor IX BIO-acetoxime is a potent dual GSK3α/β inhibitor with IC50 of 10 nM, >240-fol
R10013 PF 04691502 PF-04691502是有效和选择性的 PI3K 和 mTOR 的抑制剂。 PF-04691502与人PI3Kα,β,δ,γ和mTOR结合的 Ki 分别为1.8
R10014 AKT inhibitor VIII (Synonyms: AKTi-1/2) AKT inhibitor VIII (AKTi-1/2) 是一种细胞渗透的喹喔啉化合物,能够有效的,选择性的,可逆的抑制 Akt1,Akt2 和 Akt3 的
R10027 KU-0063794 KU-0063794 是一种有效的,特异性的 mTOR 抑制剂,能够抑制 mTORC1 和 mTORC2,IC50 值均约为 10 nM。
R10040 IP-145; Duvelisib; INK1197 Duvelisib (IPI-145, INK1197) is a novel and selective PI3K δ/γ inhibitor with Ki
R10044 WZ4003 WZ4003 is a highly specific NUAK kinase inhibitor with IC50 of 20 nM and 100 nM
R10055 OSU-03012 OSU-03012 (AR-12) is a potent inhibitor of recombinant PDK-1 with IC50 of 5 μM i
R10059 Taselisib; RG-7604; GDC-0032 GDC-0032 is a potent, next-generation β isoform-sparing PI3K inhibitor targeting
R10063 TG100115; TG100115 TG100-115 is a PI3Kγ/δ inhibitor with IC50 of 83 nM/235 nM, with little effect o
R10069 GSK2126458; Omipalisib Omipalisib (GSK2126458, GSK458) is a highly selective and potent inhibitor of p1
R10070 PKI587 Gedatolisib (PF-05212384, PKI-587) is a highly potent dual inhibitor of PI3Kα, P
R10072 GSK690693 GSK690693 is a pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 2 nM/13 nM/9 nM
R10073 Apitolisib (Synonyms: GDC-0980; GNE 390; RG 7422) Apitolisib (GDC-0980; GNE 390; RG 7422) 是一种口服有效的 PI3K 和 mTOR (TORC1/2) 激酶抑制剂,抑制
R10079 GSK2636771 GSK2636771 is a potent, orally bioavailable, PI3Kβ-selective inhibitor, sensitiv
R10082 P529 Palomid 529 (P529) inhibits both the mTORC1 and mTORC2 complexes, reduces phosph
R10085 KU-55933 KU-55933 (ATM Kinase Inhibitor) is a potent and specific ATM inhibitor with IC50
R10092 TWS11 TWS119 is a GSK-3β inhibitor with IC50 of 30 nM in a cell-free assay; capable of
R10107 NVPBKM120 BKM120 (NVP-BKM120, Buparlisib) is a selective PI3K inhibitor of p110α/β/δ/γ wit
R10136 PP242 Torkinib (PP242) is a selective mTOR inhibitor with IC50 of 8 nM in cell-free as
R10146 XL765 Voxtalisib (SAR245409, XL765) is a dual inhibitor of mTOR/PI3K, mostly for p110γ
R10167 PI103 Free base PI-103 is a multi-targeted PI3K inhibitor for p110α/β/δ/γ with IC50 of 2 nM/3 nM
R10168 YM201636 YM201636 is a selective PIKfyve inhibitor with IC50 of 33 nM, less potent to p11
R10171 AZD6482 AZD6482 is a PI3Kβ inhibitor with IC50 of 10 nM, 8-, 87- and 109-fold more selec
R10172 CHIR99021 CHIR-99021 (CT99021) is a GSK-3α and GSK-3β inhibitor with IC50 of 10 nM and 6.7
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