R10093 |
VU0364439 |
VU 0364439 is a mGlu4 positive allosteric modulator (PAM), with EC50 of 19.8 nM.
|
R10149 |
替卡格雷;Ticagrelor (AZD6140; AR-C 126532XX) |
Ticagrelor (AZD6140)是可逆有口服活性的 P2Y12 受体拮抗剂,可用来治疗血小板聚集。
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R10188 |
ciproxifan; FUB359 |
Ciproxifan is a highly potent and selective histamin H3-receptor antagonist with
|
R10211 |
LY2886721 |
LY2886721 is a BACE inhibitor used for the treatment of Alzheimer's Disease. Pha
|
R10357 |
LY310762 |
LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM, having a weaker affi
|
R10381 |
Oxiracetam |
Oxiracetam, a cyclic derivative of gamma-aminobutyric acid (GABA), is used as a
|
R10433 |
Prasugrel |
Prasugrel is a thienopyridine ADP receptor (P2Y12) antagonist, used for the redu
|
R10443 |
Carvedilol; BM14190 |
Carvedilol is a non-selective beta blocker/alpha-1 blocker, used to treat conges
|
R10451 |
Ondansetron; GR38032 |
Ondansetron is a serotonin 5-HT3 receptor antagonist used mainly as an antiemeti
|
R10452 |
Tropisetron; Novaban; SDZ-ICS930 |
Tropisetron HCl is a potent and selective 5-HT3 receptor antagonist and α7-nicot
|
R10455 |
Granisetron |
Granisetron is a serotonin 5-HT3 receptor antagonist used as an antiemetic to tr
|
R10466 |
Mianserin hydrochloride |
Mianserin盐酸盐是H1受体反向激动剂,有抗抑郁活性。
|
R10522 |
Blonanserin,AD5423 |
Blonanserin is a relatively selective serotonin (5-HT)2A and dopamine D2 antagon
|
R10523 |
Aripiprazole |
Aripiprazole is a novel atypical antipsychotic drug that is reported to be a hig
|
R10533 |
Agomelatine (S-20098) |
Agomelatine (S-20098) 是一种 MT1 和 MT2 受体的特异性激动剂,对 CHO-hMT1,HEK-hMT1,CHO-hMT2,HEK-h
|
R10538 |
Carteolol hydrochloride (OPC-1085 hydrochloride) |
Carteolol hydrochloride (OPC-1085 hydrochloride) 是非选择性β肾上腺素受体阻断剂。
|
R10551 |
Escitalopram oxalate |
Escitalopram Oxalate is a selective serotonin (5-HT) reuptake inhibitor (SSRI) w
|
R10604 |
Clemizole |
Clemizole is a H1 histamine receptor antagonist.Recently, researchers have ident
|
R10698 |
J147 |
J-147是一种广谱神经保护活性苯基酰肼化合物(EC50= 60-115nM)。
|
R10717 |
NS11394 |
NS11394 is a potent and subtype-selective GABA(A) receptor-positive modulator; p
|
R10767 |
MPEP hydrochloride |
MPEP is a potent, highly selective non-competitive antagonist at the mGlu5a rece
|
R10774 |
TG6-10-1 |
TG6-10-1 是一种 EP2 拮抗剂, 低纳摩尔下有效作用于 EP2, 比作用于人 EP3, EP4 和 IP 受体选择性高 300, EP1 受体选择性高
|
R10805 |
Elacridar HCl |
Elacridar hydrochloride is a P-glycoprotein inhibitor, and has been used both in
|
R10814 |
Muscimol HBr |
Muscimol hydrobromide is a potent but toxic structural analog of g-aminobutyric
|
R10944 |
MK-801 ; Dizocilpine |
MK-801 (Dizocilpine) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist
|