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首页 > 产品展示 > Epigenetics
目录号 产品名称 产品描述
R10008 Rucaparib phosphate; AG014699; PF01367388 Rucaparib phosphate (AG-014699 phosphate) 是一种有效、可口服的 PARP 抑制剂,结合 PARP1 的Ki 为 1.4
R10010 Rucaparib; AG-014699; PF-01367388 瑞卡帕布 Rucaparib (AG014699) 是一种有效、可口服的 PARP 抑制剂,对 PARP1 的 Ki 值为 1.4
R10015 MN-64 MN-64 is a inhibitor of tankyrases, showed 6 nM potency against tankyrase 1, iso
R10023 ACY-1215 Rocilinostat (ACY-1215) is a selective HDAC6 inhibitor with IC50 of 5 nM in a ce
R10026 INCB018424; Ruxolitinib Ruxolitinib (INCB018424) is the first potent, selective, JAK1/2 inhibitor to ent
R10033 MLN8237 Alisertib (MLN8237) is a selective Aurora A inhibitor with IC50 of 1.2 nM in a c
R10034 MK8745; MK-8745 MK-8745是极光激酶抑制剂 (aurora A),IC50 值为0.6 nM。 
R10056 Tubastatin-A Tubastatin A is a potent and selective HDAC6 inhibitor withIC50 of 15 nM in a ce
R10071 SRT1720 SRT1720 is a selective SIRT1 activator with EC50 of 0.16 μM in a cell-free assay
R10096 IOX2 IOX2 is a potent inhibitor of HIF-1α prolyl hydroxylase-2 (PHD2) with IC50 of 21
R10104 PF03814735 PF-03814735 is a novel, potent and reversible inhibitor of Aurora A/B with IC50o
R10106 MS275 Entinostat (MS-275) strongly inhibits HDAC1 and HDAC3 with IC50 of 0.51 μM and 1
R10108 Olaparib (Synonyms: AZD2281; KU0059436) Olaparib (AZD2281; KU0059436) 是一种有效的 PARP 抑制剂,抑制 PARP-1 和 PARP-2 的 IC50 分别为 5 和
R10130 VX680; MK0457; Tozasertib VX-680 (Tozasertib, MK-0457) is a pan-Aurora inhibitor, mostly against Aurora A
R10131 CYT387 Momelotinib (CYT387) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 1
R10153 FG4592 Roxadustat (FG-4592) is an HIF α prolyl hydroxylase inhibitor in a cell-free ass
R10179 4SC201 Resminostat dose-dependently and selectively inhibits HDAC1/3/6 with IC50 of 42.
R10191 CI994 CI994 (Tacedinaline) is an anti-cancer drug which inhibits HDAC1 with IC50 of 0.
R10213 SGI1776 SGI-1776 free base is a novel ATP competitive inhibitor of Pim1 with IC50 of 7 n
R10220 WP1066 WP1066 is a novel inhibitor of JAK2 and STAT3 with IC50 of 2.30 μM and 2.43 μM i
R10223 GSK503 GSK503 is a potent and specific EZH2 methyltransferase inhibitor.
R10224 Sirtinol Sirtinol 是 sirtuin 的抑制剂,对 ySir2,hSIRT2 和 hSIRT2 的 IC50 值分别为 48 μM,57.7 μM 和 131
R10232 PCI24781 PCI-24781 (Abexinostat; CRA 24781) is a novel pan-HDAC inhibitor mostly targetin
R10236 BMN673 Talazoparib (BMN 673) is a novel PARP inhibitor with IC50 of 0.58 nM in a cell-f
R10237 MGCD0103 Mocetinostat (MGCD0103) is a potent HDAC inhibitor with most potency for HDAC1 w
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