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首页 > 产品展示 > Angiogenesis
目录号 产品名称 产品描述
R10001 R788; Fostamatinib Fostamatinib (R788) 是R406的活性代谢物的原药,是Syk抑制剂,IC50为41 nM。 
R10002 R406 Free base R406 (free base) is a potent Syk inhibitor with IC50 of 41 nM in a cell-free ass
R10097 GNF-2 GNF-2 is a highly selective non-ATP competitive inhibitor of Bcr-Abl, shows no a
R10124 PCI32765; Ibrutinib Ibrutinib (PCI-32765) is a potent and highly selective Brutons tyrosine kinase (
R10181 AP24534; Ponatinib Ponatinib是一种有效的,可口服的多靶点激酶抑制剂,抑制Abl,PDGFRα,VEGFR2,FGFR1 和 Src 的 IC50 分别为0.37 nM,
R10204 PF562271 PF-562271 is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of
R10205 PF573228 PF-573228 is an ATP-competitive inhibitor of FAK with IC50 of 4 nM in a cell-fre
R10334 SU6656 SU 6656 is a selective Src family kinase inhibitor with IC50 of 280 nM, 20 nM, 1
R10363 RN486 RN486 is a potent and selective BTK inhibitor with IC50 of 4 nM.
R10367 NVPTAE226 TAE226 (NVP-TAE226) is a potent FAK inhibitor with IC50 of 5.5 nM and modestly p
R10496 Dasatinib; BMS354825 Dasatinib is a novel, potent and multi-targeted inhibitor that targets Abl, Src
R10503 Nilotinib; AMN-107 Nilotinib (AMN-107) is a Bcr-Abl inhibitor with IC50 less than 30 nM in Murine m
R10677 WH-4-023 WH-4-023 is a potent and orally active Lck/Src inhibitor with IC50 of 2 nM and 6
R10831 Dasatinib monohydrate Dasatinib Monohydrate is a novel, potent and multi-targeted inhibitor that targe
R10873 CNX-774 CNX-774是口服活性的高效Btk抑制剂,IC50< 1 nM,能与活性位点上的Cys-481形成配体导向的共价键。 
R10875 Entospletinib (GS-9973) Entospletinib (GS-9973) is an orally bioavailable, selective Syk inhibitor with
R10917 Radotinib; IY-5511 Radotinib (IY-5511) 是酪氨酸激酶 Bcr-Abl1 新型选择性抑制剂,对野生型 Bcr-Abl1 的 IC50 值为 34nM。 
R10967 PF-431396 PF-431396 is a dual PYK2/FAK inhibitor with IC50 of 11 nM and 2 nM, respectively
R10997 GNF-7 GNF-7 is a potent type-II kinase Bcr-Abl inhibitor with IC50 of <5 nM, 61 nM, 12
R11448 Fostamatinib Disodium (Synonyms: R788(Disodium)) Fostamatinib Disodium (R788 Disodium) 是活性代谢物R406的原药,是Syk抑制剂,IC50为41 nM。 
R11633 GZD824 (Synonyms: HQP1351) GZD824 (HQP1351) 是可口服的 Bcr-Abl 抑制剂,对野生型和 T315I 突变型 IC50 分别为 0.34 和 0.68 nM。
R11585 BAY-61-3606 BAY-61-3606 is a potent and selective inhibitor of Syk kinase (Ki = 7.5 nM).
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