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R10016 TH287 TH287是MTH1 (NUDT1)高效选择性抑制剂,IC50值0.8nM,对MTH2, NUDT5, NUDT12, NUDT14等抑制力弱。
R10019 Setanaxib (Synonyms: GKT137831; GKT831) Setanaxib (GKT137831) 是选择性的NADPH氧化酶 (NOX1/4) 抑制剂,Ki 分别为140和110nM。 
R10020 JNJ-31020028 JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 recept
R10024 Cardiogenol C hydrochloride Cardiogenol C盐酸盐是一种细胞渗透性的嘧啶化合物, 有效诱导胚胎干细胞分化为心肌 (EC50= 100 nM)。 
R10030 MLN4924 MLN4924 is a potent and selective small molecule NEDD8-activating enzyme (NAE) i
R10041 Vesnarinone (OPC-8212) Vesnarinone是一种喹啉酮衍生物, 药效学效应包括抑制磷酸二酯酶III (PDE3) 活性,增加钙通量, 及减小钾通量。 
R10045 Fluoroclebopride
R10047 Vortioxetine Vortioxetine (Lu AA21004) is a multimodal serotonergic agent, inhibits 5-HT1A, 5
R10048 Temsavir; BMS-626529 BMS-626529 is a novel small-molecule attachment inhibitor that targets HIV-1 gp1
R10049 TP-808;TP808 TP808是影响多种四环素抗生素合成的关键中间体。
R10060 Nadifloxacin; Acuatim; Nadixa; OPC7251 Nadifloxacin is a topical fluoroquinolone antibiotic for the treatment of acne v
R10080 TH-302 TH-302 is selective hypoxia-activated prodrug targeting hypoxic regions of solid
R10081 TAS103 dihydrochloride TAS-103 2Hcl(BMS-247615 2Hcl) is a dual inhibitor of topoisomerase-I (topo-I) an
R10084 Orteronel; TAK-700 Orteronel(TAK-700) was selected as a candidate for clinical evaluation. orterone
R10086 BAY571293 Pritelivir (BAY 57-1293) is a potent helicase primase inhibitor, exhibiting anti
R10088 RTA408; Omaveloxolone RTA-408 是一种抗氧化炎症调节剂 (AIM),可激活 Nrf2 并抑制一氧化氮 (NO)。RTA-408 通过抑制 STING 依赖的
R10102 AKR501 Avatrombopag(AKR-501; AS1670542) is a novel orally-active thrombopoietin(TPO) re
R10105 Nelfinavir Nelfinavir(AG-1341) is a potent and orally bioavailable human immunodeficiency v
R10122 Nitisinone Nitisinone(SC0735) is an inhibitor of the enzyme 4-hydroxyphenylpyruvate dioxyge
R10137 AP23464
R10145 ABT102
R10147 LY335979 Zosuquidar (LY335979) is a potent modulator of P-glycoprotein-mediated multi-dru
R10154 CTP518
R10155 Posaconazole; SCH56592; Noxafil Posaconazole 是一种广谱的,二代三唑类物质,具有抗真菌作用。 
R10164 Avibactam sodium; NXL-104 阿维巴坦钠 Avibactam sodium (NXL-104) 是一种共价,可逆的非β-内酰胺 β-内酰胺酶抑制剂 (β-lactamase) 抑制剂,抑制
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