R10184 |
GW9508 |
GW9508 is a potent and selective agonist for FFA1 (GPR40) with pEC50 of 7.32, 10
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R10194 |
OC000459 |
OC000459 is a potent and selective D prostanoid receptor 2 (DP2) antagonist with
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R10244 |
Fasiglifam (TAK-875) |
Fasiglifam (TAK-875) 是一种有效的,可口服的,具有选择性的 GPR40 激动剂,EC50 值为 72 nM。
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R10415 |
AZD1981 |
AZD1981 is a potent, selective CRTh2 (DP2) receptor antagonist with IC50 of 4 nM
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R10674 |
APD668 |
APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and
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R10893 |
JNJ38431055; APD-597 |
APD597是GPR119激动剂, 作用于hGPR119, EC50为46 nM, 可用于治疗2型糖尿病。
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