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目录号 产品名称 产品描述
R10083 XL413 Hydrochloride XL413 hydrochloride 是一种有效的,选择性的,ATP 竞争性的 Cdc7 抑制剂,IC50 值为 3.4 nM,同时对 CK2 和 PIM1
R10090 AZD5438 AZD-5438 是有效的 CDK1/2/9 抑制剂,IC50 值分别为 16 nM/6 nM/20 nM;对GSK3β,CDK5,CDK6的抑制作用较弱。&n
R10139 Roscovitine; Seliciclib Roscovitine (Seliciclib, CYC202) is a potent and selective CDK inhibitor for Cdc
R10189 AT7519 HCl AT7519 HCl is a multi-CDK inhibitor for CDK1, 2, 4, 6 and 9 with IC50 of 10-210
R10314 PD0332991; PD0332991; Palbociclib Palbociclib (PD0332991) Isethionate is a highly selective inhibitor of CDK4/6 wi
R10341 BS-181 hydrochloride BS-181盐酸盐是CDK7高效选择性抑制剂,IC50值21nM,对CDK1/92/4/5/6/9作用弱。 
R10377 Palbociclib hydrochloride;PD 0332991 hydrochloride Palbociclib hydrochloride是高选择性的 CDK4/6 抑制剂,IC50 分别为11 nM 和 16 nM。 
R10707 PURVALANOLA Purvalanol A is a potent, and cell-permeable CDK inhibitor with IC50 of 4 nM, 70
R10729 BML-277 BML-277 (Chk2 Inhibitor II) is a Chk2 (checkpoint kinase 2) inhibitor.
R10755 BPR1J-097 BPR1J-097 是一个新型且强效的 FLT3 抑制剂,其 IC50 值为 11 nM。
R10910 MK-8776 MK-8776 (SCH 900776) is a selective Chk1 inhibitor with IC50 of 3 nM in a cell-f
R11449 AT7519 AT7519 是一种有效的 CDK 抑制剂,对 CDK1,CDK2,CDK4-CDK6 以及 CDK9 的 IC50 值分别为 210,47,100,13,17
R11461 Abemaciclib methanesulfonate (LY2835219 methanesulfonate) Abemaciclib methanesulfonate (LY2835219 methanesulfonate) 是选择性的 CDK4/6 
R11611 KENPAULLONE Kenpaullone is an ATP-competitive inhibitor of cyclin-dependent kinases (CDKs).
R11620 Ro 3306 RO-3306 is an ATP-competitive, and selective CDK1 inhibitor with Ki of 20 nM, >1
R2032672 PHA767491 PHA-767491 是一种 Cdc7-Dbf4 (DDK)/Cdk9 的双重抑制剂,IC50 值分别为 10 nM 和 34 nM。
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