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首页 > 产品展示 > Metabolism
目录号 产品名称 产品描述
R10091 LCZ696;Sacubitril;Valsartan Varespladib (LY315920) 是一种有效且具有选择性的 group IIA, secretory phospholipase A2 (sPLA2
R10112 Abiraterone Acetate; CB7630 Abiraterone acetate 是一种口服、有效、选择性和不可逆的 CYP17A1 抑制剂,具有抗雄激素活性。Abiraterone acetate是
R10113 Abiraterone; CB7598 Abiraterone is a potent CYP17 inhibitor with IC50 of 2 nM in a cell-free assay.
R10120 Bexarotene Bexarotene is a retinoid specifically selective for retinoid X receptors, used a
R10125 TOK001; VN1241 Galeterone is a selective CYP17 inhibitor and androgen receptor (AR) antagonist
R10159 Anacetrapib; MK0859 Anacetrapib 是一种有效的 CETP 抑制剂,作用于 rhCETP 和 C13S CETP 突变型,IC50 分别为 7.9±2.5 nM 和 11.
R10162 Apremilast; CC10004 Apremilast (CC-10004) is a potent and orally active PDE4 and TNF-α inhibitor wit
R10209 indisulam; E7070 Indisulam (E7070) is a carbonic anhydrase inhbitor, is also a novel synthetic su
R10344 GW9662 GW9662 is a selective PPAR antagonist for PPARγ with IC50 of 3.3 nM in a cell-fr
R10432 Rivaroxaban; Xarelto; BAY 59-7939 Rivaroxaban is a direct inhibitor of Factor Xa with Ki and IC50 of 0.4 nM and 0.
R10444 Olprinone Olprinone(Loprinone) is a selective phosphodiesterase 3 (PDE3) inhibitor.
R10456 Gimeracil Gimeracil is an inhibitor of dihydropyrimidine dehydrogenase, which inhibits the
R10482 Tadalafil Tadalafil is a PDE-5 inhibitor with IC50 of 1.8 nM in a cell-free assay.
R10485 Epacadostat (Synonyms: INCB 024360) Epacadostat (INCB 024360) 是一种有效,选择性的 IDO1 抑制剂, IC50 为 71.8 nM±17.5 nM。 
R10526 Anagrelide hydrochloride; BL4162A Anagrelide is a drug used for the treatment of essential thrombocytosis.
R10570 Safinamide mesylate Safinamide Mesylate is mesylate salt of Safinamide, selectively and reversibly i
R10591 NSC14613; PluriSln1 PluriSIn1 is an inhibitor of the stearoyl-coA desaturase 1 (SCD1), which is able
R10632 AGI-6780 AGI-6780 is a potent, selective inhibitor of mutant IDH2 with an IC50 value of 2
R10648 Dimethyloxaloylglycine;DMOG DMOG is an antagonist of α-ketoglutarate cofactor and inhibitor for HIF prolyl h
R10659 Fenretinide; 4-HPR Fenretinide is a synthetic retinoid agonist. It is an antiproliferative, antioxi
R10724 Moclobemide Moclobemide is a MAO-A (5-HT) inhibitor with IC50 of 6.1 μM.
R10735 U-104 U-104是碳酸酐酶(Carbonic anhydrase)CA IX和CA XII高效抑制剂,Ki值分别为45.1nM和4.5nM。
R10801 Deltarasin Deltarasin is a small molecular inhibitor of KRAS-PDEδ interaction with Kd of 38
R10665 IDO-IN-7;NLG-919 analogue; GDC-0919 analogue IDO-IN-7 (NLG-919 analogue) 是一种有效的 IDO1 抑制剂, IC50为 38 nM。 
R10842 Mycophenolate mofetil; Linfonex Mycophenolate Mofetil is a non-competitive, selective and reversible inhibitor o
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