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首页 > 产品展示 > GPCR & G Protein
目录号 产品名称 产品描述
R10066 Dapagliflozin; BMS512148 Dapagliflozin (BMS-512148) 是一种用于治疗糖尿病 (DM) 的新型药物,是一种竞争性葡萄糖协同转运蛋白2 (SGLT2) 抑制剂,可导
R10123 Bosetan Bosentan is an endothelin (ET) receptor antagonist for ET-A and ET-B with Ki of
R10132 Canagliflozin Canagliflozin is a highly potent and selective SGLT2 inhibitor for hSGLT2 with I
R10185 Otenabant Hydrochloride (CP 945598 Hydrochloride) Otenabant (CP945598)盐酸盐是CB1受体高亲和性拮抗剂,Ki为0.7 nM。
R10186 CP945598 free base Otenabant 是一种有效的,选择性的 cannabinoid receptor CB1 拮抗剂,Ki 值为 0.7 nM,对其选择性是对 CB2 的 10
R10242 AMG073 Cinacalcet HCl represents a new class of compounds for the treatment of hyperpar
R10260 Sotagliflozin; LP802034; LX4211 Sotagliflozin (LX-4211) 是SGLT1/2抑制剂,是抗糖尿病剂。 
R10406 AMD3465 hexahydrobromide (GENZ-644494 hexahydrobromide) AMD 3465 hexahydrobromide (GENZ-644494 hexahydrobromide) 是一种有效的 CXCR4 拮抗剂,在 SupT
R10436 Ambrisentan; BSF208075; LU208075 Ambrisentan 是一种选择性的ET A型受体 (ETAR) 拮抗剂。 
R10488 Empagliflozin Empagliflozin是一种选择性钠葡萄糖协同转运蛋白-2 (SGLT-2) 抑制剂,抑制人SGLT-2的IC50 为3.1 nM。 
R10489 Canagliflozin hemihydrate Canagliflozin 0.5 H2O(JNJ 28431754; TA 7284) is a highly potent and selective SG
R10491 Ipragliflozin Ipragliflozin (ASP1941) is a highly potent and selective SGLT2 inhibitor with IC
R10492 Tofogliflozin Tofogliflozin(CSG-452) hydrate is a potent and highly specific sodium/glucose co
R10543 Plerixafor; AMD310 Plerixafor (AMD3100) is a chemokine receptor antagonist for CXCR4 and CXCL12-med
R10609 Reversine Reversine 是一种ATP-竞争性的 Aurora kinase 抑制剂,作用于 Aurora A,Aurora B 和 Aurora C,IC50 分别
R10725 CYM5442 CYM 5442 HCl is a potent and selective EDG-1 (S1P1) agonist in vitro (EC50 = 1.3
R10794 Capadenoson; BAY 68-4986 Capadenoson (BAY 68-4986) is a new adenosine A1 receptor agonist.
R10848 Ki16198 Ki16198 is the methyl ester of Ki16425, which is a LPA antagonist and inhibits L
R10950 ozanimod;RPC1063;RPC-1063 Ozanimod 是一种有效的选择性 S1P1 和 S1P5 受体激动剂,在[35S]-GTPγS 结合实验中,EC50 分别为 410±160 pM 和 11
R10953 ABC294640 ABC294640 is an orally bioavailable and selective sphingosine kinase-2 (SphK2) i
R11455 Plerixafor octahydrochloride; AMD3100 octahydrochloride; JM3100 octahydrochloride; SID791 octahydrochloride Plerixafor octahydrochloride (AMD3100 octahydrochloride) 是一种选择性的 CXCR4 
R11505 SQ22536 SQ22536 is an inhibitor of adenylyl cyclase with an IC50 of 1.4 μM. It can inhib
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