R2101028 |
Nisoxetine hydrochloride |
Nisoxetine hydrochloride 是一种有效的和选择性的去甲肾上腺素转运蛋白 (NET) 的抑制剂,Kd 值为 0.76 nM。Nisoxeti
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R2101029 |
ASN03576800 |
ASN03576800 is an inhibitor of the VP40 matrix protein.
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R2101030 |
HA-155 |
HA155 (Autotaxin Inhibitor IV), a boronic acid-based compound, inhibits autotaxi
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R2101031 |
CYM5520 |
noncompetitive allosteric agonist of S1P2
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R2101032 |
CRT5 |
CRT5 (CRT0066051), a pyrazine benzamide, is a potent and selective PKD inhibitor
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R2101033 |
BMS453 |
BMS453 (BMS-189453) 是一种合成类维生素 A,是一种 RARβ 激动剂和 RARα/RARγ 拮抗剂。BMS453 主要通过诱导活性 TGFβ
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R2101034 |
Mps1-IN-3 |
Mps1-IN-3 是一种有效的,选择性的 MPS1 抑制剂,IC50 值为 50 nM。
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R2101035 |
OS-3-106 |
OS-3-106 is a novel dopamine D3 receptor-selective partial agonist.
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R2101036 |
NSC-703786 |
A potent, selective antitumour agent through activation the aryl hydrocarbon rec
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R2101037 |
GW779439X |
GW779439X is an inhibitor of cyclin dependent kinase.
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R2101038 |
RO2959 hydrochloride |
RO2959 hydrochloride 是一种有效的选择性 CRAC 通道抑制剂,IC50 为 402 nM。RO2959 hydrochloride 是由
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R2101039 |
Flupenthixol dihydrochloride |
cis-(Z)-Flupentixol dihydrochloride 是有效、选择性的多巴胺DA D1/D2 受体的拮抗剂,其对D2 受体和 5-HT2A 的
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R2101040 |
4BP-TQS |
4BP-TQS is an allosteric agonist of α7 subunit-containing neuronal nicotinic ace
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R2101041 |
B355252 |
B355252 is a neuroprotective agent that potentiates nerve growth factor (NGF)-in
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R2101042 |
GSK 2830371 |
GSK 2830371 是一种选择性的Wip1磷酸酶 (Wip1 phosphatase)抑制剂,IC50 为 6 nM。
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R2101043 |
MONNA |
MONNA is a potent TMEM16A (Anoctamin-1) blocker (IC50 = 80 nM). Exhibits >100
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R2101044 |
TAE-1 |
TAE-1 is an inhibitor of amyloid-β fibril formation and aggregation, suggesting
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R2101045 |
ML191 |
ML-191 is a potent, selective GPR55 antagonist with 160 nM potency for GPR55 and
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R2101046 |
ML336 |
ML-336 is an inhibitor of of the Venezuelan equine encephalitis virus (VEEV) str
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R2101047 |
GW280264X |
GW280264X is an ADAM17 inhibitor.
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R2101048 |
TM5007 |
TM5007 is a poent inhibitor plasminogen activator inhibitor-1 (PAI-1) with IC50
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R2101049 |
CYM2503 |
CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that poten
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R2101050 |
YM26734 |
YM-26734 is a rabbit platelet sPLA2 inhibitor that has been used to ameliorate l
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R2101051 |
G244-LM |
G244-LM is a potent and specific tankyrase 1/2 inhibitor that inhibits Wnt signa
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R2101052 |
VK-II-86 |
VK-II-86 is a selective ryanodine receptor type 2 (RyR2) antagonist.
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