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目录号 产品名称 产品描述
R10211 LY2886721 LY2886721 is a BACE inhibitor used for the treatment of Alzheimer's Disease. Pha
R10213 SGI1776 SGI-1776 free base is a novel ATP competitive inhibitor of Pim1 with IC50 of 7 n
R10214 LY411575; YO01027 YO-01027 (Dibenzazepine) is a dipeptidic γ-secretase inhibitor with IC50 of 2.6
R10216 PLX4032 Vemurafenib (PLX4032, RG7204) is a novel and potent inhibitor of B-RafV600E with
R10219 AZD7762;AZD-7762 AZD-7762 是一种有效的ATP竞争性的细胞周期检测点激酶 (checkpoint kinase,Chk) 抑制剂,抑制Chk1的 IC50&nb
R10224 Sirtinol Sirtinol 是 sirtuin 的抑制剂,对 ySir2,hSIRT2 和 hSIRT2 的 IC50 值分别为 48 μM,57.7 μM 和 131
R10225 LY-364947 (HTS466284) Y-364947 是一种有效的,ATP 竞争性的 TGFβR-I 抑制剂,IC50 值为 59 nM,是对 TGFβR-II 选择性的 7 倍。 
R10227 TAK438; Vonoprazan Fumarate Vonoprazan Fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid block
R10233 Tyrphostin A9;Tyrphostin 9; Malonoben Tyrphostin A9 是51种酪氨酸激酶抑制剂,是线粒体分裂诱导剂。 
R10235 GSK1838705A GSK1838705A是高效,可逆的 IGF-IR 和胰岛素受体 (insulin receptor) 抑制剂,IC50 值分别为
R10236 Talazoparib (BMN 673) Talazoparib (BMN-673) 是高效的 PARP1/2 抑制剂,Ki 值分别为 1.2 nM 和 0.87 nM。 
R10239 Tubastain A Tubastatin A is a potent and selective HDAC6 inhibitor with IC50 of 15 nM in a c
R10242 AMG073 Cinacalcet HCl represents a new class of compounds for the treatment of hyperpar
R10243 GDC0941; Pictilisib Pictilisib (GDC-0941) is a potent inhibitor of PI3Kα/δ with IC50 of 3 nM in cell
R10244 Fasiglifam (TAK-875) Fasiglifam (TAK-875) 是一种有效的,可口服的,具有选择性的 GPR40 激动剂,EC50 值为 72 nM。
R10245 Ostarine; MK2866 Andarine is a selective non-steroidal androgen receptor (AR) agonist with Ki of
R10246 司马西特;Semagacestat (LY450139) Semagacestat 是一种 γ-secretase 抑制剂,抑制 β-amyloid (Aβ42),Aβ38&nb
R10247 Veliparib dihydrochloride; ABT-888 dihydrochloride Veliparib dihydrochloride是有效的 PARP1 和 PARP2 抑制剂,Ki 分别为5.2 nM,2.9 nM。 
R10248 NSC713200 Bardoxolone Methyl is an IKK inhibitor, showing potent proapoptotic and anti-inf
R10250 TAK632 TAK-632 is a potent pan-Raf inhibitor with IC50 of 8.3 nM and 1.4 nM for B-Raf(w
R10251 BMS232632; CGP73547; HSDB7339; Atazanavir Sulfate is a HIV protease inhibitor with Ki of 2.66 nM in a cell-free
R10252 MK1775 MK-1775 is a potent and selective Wee1 inhibitor with IC50 of 5.2 nM in a cell-f
R10253 Dacomitinib,PF299804 Dacomitinib 是一种特异,不可逆的 ERBB 家族抑制剂,作用于 EGFR,ERBB2 和 ERBB4 的 IC50 分别为 6 nM,45.7 nM
R10254 AZD9291 Mesylate Osimertinib mesylate (AZD-9291 mesylate) 是不可逆的突变体选择性 EGFR 抑制剂;对EGFRL858R 和EGFRL8
R10255 LY2874455; dovitinib LY2874455 is a pan-FGFR inhibitor with IC50 of 2.8 nM, 2.6 nM, 6.4 nM, and 6 nM
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