电话: | 021-31433387 |
15618786686(微信) | |
Email: | sales@rechemscience.com |
info@rechemscience.com | |
QQ: | 1369748377 |
Skype: | rechem@outlook.com |
目录号 | 产品名称 | 产品描述 |
R10211 | LY2886721 | LY2886721 is a BACE inhibitor used for the treatment of Alzheimer's Disease. Pha |
R10213 | SGI1776 | SGI-1776 free base is a novel ATP competitive inhibitor of Pim1 with IC50 of 7 n |
R10214 | LY411575; YO01027 | YO-01027 (Dibenzazepine) is a dipeptidic γ-secretase inhibitor with IC50 of 2.6 |
R10216 | PLX4032 | Vemurafenib (PLX4032, RG7204) is a novel and potent inhibitor of B-RafV600E with |
R10219 | AZD7762;AZD-7762 | AZD-7762 是一种有效的ATP竞争性的细胞周期检测点激酶 (checkpoint kinase,Chk) 抑制剂,抑制Chk1的 IC50&nb |
R10224 | Sirtinol | Sirtinol 是 sirtuin 的抑制剂,对 ySir2,hSIRT2 和 hSIRT2 的 IC50 值分别为 48 μM,57.7 μM 和 131 |
R10225 | LY-364947 (HTS466284) | Y-364947 是一种有效的,ATP 竞争性的 TGFβR-I 抑制剂,IC50 值为 59 nM,是对 TGFβR-II 选择性的 7 倍。 |
R10227 | TAK438; Vonoprazan Fumarate | Vonoprazan Fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid block |
R10233 | Tyrphostin A9;Tyrphostin 9; Malonoben | Tyrphostin A9 是51种酪氨酸激酶抑制剂,是线粒体分裂诱导剂。 |
R10235 | GSK1838705A | GSK1838705A是高效,可逆的 IGF-IR 和胰岛素受体 (insulin receptor) 抑制剂,IC50 值分别为 |
R10236 | Talazoparib (BMN 673) | Talazoparib (BMN-673) 是高效的 PARP1/2 抑制剂,Ki 值分别为 1.2 nM 和 0.87 nM。 |
R10239 | Tubastain A | Tubastatin A is a potent and selective HDAC6 inhibitor with IC50 of 15 nM in a c |
R10242 | AMG073 | Cinacalcet HCl represents a new class of compounds for the treatment of hyperpar |
R10243 | GDC0941; Pictilisib | Pictilisib (GDC-0941) is a potent inhibitor of PI3Kα/δ with IC50 of 3 nM in cell |
R10244 | Fasiglifam (TAK-875) | Fasiglifam (TAK-875) 是一种有效的,可口服的,具有选择性的 GPR40 激动剂,EC50 值为 72 nM。 |
R10245 | Ostarine; MK2866 | Andarine is a selective non-steroidal androgen receptor (AR) agonist with Ki of |
R10246 | 司马西特;Semagacestat (LY450139) | Semagacestat 是一种 γ-secretase 抑制剂,抑制 β-amyloid (Aβ42),Aβ38&nb |
R10247 | Veliparib dihydrochloride; ABT-888 dihydrochloride | Veliparib dihydrochloride是有效的 PARP1 和 PARP2 抑制剂,Ki 分别为5.2 nM,2.9 nM。 |
R10248 | NSC713200 | Bardoxolone Methyl is an IKK inhibitor, showing potent proapoptotic and anti-inf |
R10250 | TAK632 | TAK-632 is a potent pan-Raf inhibitor with IC50 of 8.3 nM and 1.4 nM for B-Raf(w |
R10251 | BMS232632; CGP73547; HSDB7339; | Atazanavir Sulfate is a HIV protease inhibitor with Ki of 2.66 nM in a cell-free |
R10252 | MK1775 | MK-1775 is a potent and selective Wee1 inhibitor with IC50 of 5.2 nM in a cell-f |
R10253 | Dacomitinib,PF299804 | Dacomitinib 是一种特异,不可逆的 ERBB 家族抑制剂,作用于 EGFR,ERBB2 和 ERBB4 的 IC50 分别为 6 nM,45.7 nM |
R10254 | AZD9291 Mesylate | Osimertinib mesylate (AZD-9291 mesylate) 是不可逆的突变体选择性 EGFR 抑制剂;对EGFRL858R 和EGFRL8 |
R10255 | LY2874455; dovitinib | LY2874455 is a pan-FGFR inhibitor with IC50 of 2.8 nM, 2.6 nM, 6.4 nM, and 6 nM |