R2101103 |
Farampator (CX-691;Org24448) |
Farampator (CX-691;Org24448) 是一种AMPA受体正调节剂。
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R2101104 |
GSK3 Inhibitor XIII |
GSK3 Inhibitor XIII (GSK3i XIII) is an ATP-binding site inhibitor of GSK-3.
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R2101105 |
pythiDC |
PythiDC is a selective inhibitor of collagen prolyl 4-hydroxylase.
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R2101106 |
(S)SHA-68 |
SHA-68 is a selective neuropeptide S receptor (NPSR) antagonist that displays no
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R2101107 |
NCGC607 |
NCGC607 is a a small-molecule noninhibitory chaperone of glucocerebrosidase.
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R2101108 |
ML266 (CID-46943215) |
ML266 (CID-46943215) is a activator of glucocerebrosidase (GCase) that does not
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R2101109 |
BMS986187 |
BMS-986187 is a novel potent, positive allosteric modulator of δ-opioid receptor
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R2101110 |
BMS986188 |
BMS-986188 is a positive allosteric modulator (PAM) of δ-opioid receptors with E
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R2101111 |
R243 |
R243是一种有效的小分子CCR8拮抗剂,可抑制CCR8信号传导和趋化性,抑制CCL1诱导的Ca2+通量和CCL1驱动的腹膜巨噬细胞在0.2μM时聚集;减弱TN
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R2101112 |
BGC-20-1531 |
BGC-20-1531 is a EP4 antagonist for the treatment of acute migraine.
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R2101113 |
Aka Lumine |
AkaLumine is a luciferin analogue. The bioluminescence produced by AkaLumine in
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R2101114 |
SGC2085 hydrochloride |
SGC2085 is a potent and selective coactivator associated arginine methyltransfer
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R2101115 |
TMP778 |
TMP778 是一种有效的、RORγt 的选择性反向激动剂,其 FRET 检测出的 IC50 值为 7 nM。
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R2101116 |
TX1-85-1 |
TX1-85-1 是一种 Her3 (ErbB3) 抑制剂,IC50 值为 23 nM。TX1-85-1 可诱发 Her3 蛋白的部分降解并减弱 Her3 依赖
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R2101117 |
Azaindole 1;TC-S 7001 |
Azaindole 1 是一种高效的人 ROCK-1 和 ROCK-2 抑制剂,IC50 值分别为 0.6 和 1.1 nM,同时可抑制小鼠和大鼠 ROCK-2
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R2101118 |
Shield-1 |
Shield-1 是特异性,细胞可渗透的,高亲和力 FK506 结合蛋白-12 (FKBP) 配体,通过与突变的 FKBP (mtFKBP) 结合而逆转其不稳定
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R2101119 |
NCGC00262650 |
NCGC00262650 is a dual inhibitor of AMA1-RON2 interaction and c-Src tyrosine kin
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R2101120 |
ERDRP-0519 |
ERDRP-0519 is an orally available polymerase inhibitor. It shows efficacy agains
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R2101121 |
AQX-016A |
AQX-016A is a potent activator of SHIP-1 that induces apoptosis of the cancer ce
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R2101122 |
WWL229 |
WWL229 is a selective Ces3 inhibitor. It acts by inhibiting recombinant Ces3 but
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R2101123 |
KLH45 |
KLH45 is a selective inhibitor of DDHD2 (DDHD domain containing 2).
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R2101124 |
AA 41612 |
AA 41612 is a potent, synthetic melanopsin antagonist with IC50 of 15.8 nM, atte
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R2101125 |
ML-349 |
ML349 是一个有效且特异的酰基蛋白硫酯酶 2 (APT-2) 抑制剂,其 Ki 值为 120 nM。ML349 也是 LYPLA2 的抑制剂,其 IC50
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R2101126 |
GNE-140 racemate |
GNE-140外消旋体是一种新型高效乳酸脱氢酶(LDHA)抑制剂。在MIA-PaCa-2人胰腺细胞中,LDHA抑制迅速影响了整体代谢,但细胞死亡只发生在持续抑制
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R2101127 |
Soporidine |
Soporidine is a strigolactone (SL) antagonist and inhibitor of germination in th
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