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产品展示
目录号
产品名称
产品描述
R2031168
(R)-N-(pyrrolidin-3-ylmethyl)methanesulfonamide
该产品曾做过需定制
R2030218
Pristinamycin IA (Mikamycin B;Mikamycin IA)
Pristinamycin IA (Mikamycin B;Mikamycin IA) 是一个环肽大环内酯抗生素,属于 链霉杀阳菌素,也是P-glycoprot
R2003041
LIT-001 TFA
LIT-001 是第一种非肽类催产素受体 (OT-R) 激动剂 (EC50=55 nM; Ki=226 nM)。LIT-001 改善孤独症小鼠模型的社交互动。&
R2003051
Cefminox sodium (MT-141)
Cefminox sodium (MT-141) 是一种半合成的头霉素,具有广谱的抗菌活性。Cefminox sodium (MT-141) 为前列环素受体 (
R2003081
SRT3025 HCl;Sirtuin modulator 1
Sirtuin modulator 1 是 SIRTl (SIRT3 的同系物) 的调节剂,EC1.5 值 < 1 μM,摘自专利 WO 20100718
R00391
沙芬酰胺;Safinamide (FCE 26743)
沙芬酰胺 Safinamide (FCE 26743)是可逆的 MAO-B 抑制剂,IC50 为 98 nM,比对 MAO-A 的抑制性高5918 倍。&nbs
R00310
Nilotinib Impurity 9
Nilotinib是一种口服可用的具有抗肿瘤活性的 Bcr-Abl 酪氨酸激酶抑制剂。
R00311
Cardiogenol C, Hydrochloride
Cardiogenol C盐酸盐是一种细胞渗透性的嘧啶化合物, 有效诱导胚胎干细胞分化为心肌 (EC50= 100 nM)。
R00313
Cisplatin (CDDP; cis-Diaminodichloroplatinum)
Cisplatin 是一种抗肿瘤化疗药物,它与 DNA 交联引起癌细胞中DNA损伤。
R00314
Defactinib (VS-6063, PF-04554878)
Defactinib (VS-6063; PF-04554878) 是一种新型 FAK 抑制剂,抑制 FAK 在 Tyr397 位点磷酸化,这种作用具有时间和剂
R00315
Defactinib hydrochloride;VS-6063 hydrochloride; PF 04554878 hydrochloride
Defactinib hydrochloride (VS-6063 hydrochloride; PF 04554878 hydrochloride) 是一种新
R00318
Donepezil;E2020 free base
Donepezil (E2020 free base) 是 AChE 抑制剂,对 bAChE 和 hAChE 的 IC50 分别为 8.12 nM 和 11.6
R00320
Olodaterol Hydrochloride
Olodaterol hydrochloride是Olodaterol的盐酸盐形式,Olodaterol是一种长效的β2肾上腺素能受体(beta2-adrene
R00321
RET-IN-1
RET-IN-1是一种有效的 RET 激酶抑制剂,抑制 RET (WT),RET (V804M) 和 RET (G810R),IC50&nb
R2030453
Ethyl 4-(1-hydroxy-1-methylethyl)-2-propyl-imidazole-5-carboxylate
R2030454
ETHYL 1,5-DIMETHYL-1H-PYRAZOLE-3-CARBOXYLATE
R2030455
(2S)-2-AMino-2-(3-chlorophenyl)ethan-1-ol
R2030456
4-(5-chloro-2-isopropylaminopyridin-4-yl)-1-(toluene-4-sulfonyl)-1H-pyrrole-2-carboxylic acid methyl ester
R2030457
4-(5-chloro-2-(isopropylaMino)pyridin-4-yl)-1H-pyrrole-2-carboxylic acid
NA.
R2030458
Ulixertinib hydrochloride (BVD-523 hydrochloride; VRT752271 hydrochloride)
Ulixertinib hydrochloride (BVD-523 hydrochloride) 是一种有效、可口服、高度选择性、ATP-竞争性、可逆、共价的
R2030459
2-Chloro-6-methylnicotinic acid
R2030460
3-(2-methoxy-6-methylpyridin-3-yl)-1H-pyrazol-5-amine
R2030461
tert-butyl(R)-3-((6-chloropyrazin-2-yl)oxy)piperidine-1-carboxylate
R2030462
1,2,3-cyclopropanetri-carboxylic acid
R2032111
ALK2-IN-1;BLU782
ALK2-IN-1 是一种活化素受体样激酶 2 (ALK2) 抑制剂,IC50<10 nM。详细信息请参考专利文献 WO2017181117A1 中的化合
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