R10764 |
BMH-21 |
BMH-21 is a DNA intercalator, which binds ribosomal DNA and inhibits RNA polymer
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R10766 |
SC-202671 |
JNK inhibitor IX is a selective and potent JNK inhibitor with pIC50 of 6.5 and 6
|
R10767 |
MPEP hydrochloride |
MPEP is a potent, highly selective non-competitive antagonist at the mGlu5a rece
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R10768 |
KU-60019 |
KU-60019 is an improved analogue of KU-55933, with IC50 of 6.3 nM for ATM in cel
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R10769 |
O4I2 |
O4I2 is a potent Oct3/4 inducer in various human cell lines including human fibr
|
R10771 |
O4I1 |
O4I1 is as a potent Oct3/4 inducer.Target: Oct3/4
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R10774 |
TG6-10-1 |
TG6-10-1 是一种 EP2 拮抗剂, 低纳摩尔下有效作用于 EP2, 比作用于人 EP3, EP4 和 IP 受体选择性高 300, EP1 受体选择性高
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R10775 |
B7/CD28 interaction inhibitor 1 |
B7/CD28 interaction inhibitor 1 (copmound 6b) 是一种有效的 B7.1-CD28 相互作用抑制剂,IC50 为 50
|
R10776 |
4-Keto13-cis-Retinoic Acid |
|
R10778 |
Pimelic diphenylamide 106; TC-H106 |
Pimelic diphenylamide 106 is a slow, tight-binding inhibitor of class I HDAC (HD
|
R10779 |
UF010 |
UF010是一种有效的选择性HADC抑制剂, 作用于HDACs 3, 2, 1 和 8, IC50值分别为 0.06μM, 0.1μM, 0.5μM, 和1.5
|
R10780 |
KC7F2 |
KC7F2 是一种有效的缺氧诱导因子 HIF-1 通道抑制剂,在 LN229-HRE-AP 细胞中 IC50 值为 20 μM,可用作癌症治疗剂。
|
R10781 |
WDR50103 |
WDR5-0103 is a potent and selective WD repeat-containing protein 5 (WDR5) antago
|
R10782 |
Losartan Carboxylic Acid (E-3174) |
Losartan Carboxylic Acid (E-3174) 是 Losartan 的活性羧酸代谢产物,是血管紧张素 Ⅱ 受体 1 型 (AT1
|
R10783 |
vorapaxar intermediate 1 |
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R10784 |
vorapaxar intermediate 2 |
|
R10785 |
Savolitinib (Volitinib; HMPL-504; AZD-6094) |
volitinib (AZD-6094) 是一种高效选择性、口服生物利用度 c-Met 抑制剂,对 c-Met 和 p-Met 的 IC50 分别为 5 nM
|
R10786 |
FMK |
FMK is a RSK2 kinase inhibitor.
|
R10789 |
CPI-203 |
CPI203 is a novel potent, selective and cell permeable inhibitor of the bromodom
|
R10790 |
2-(2,6-dimethylphenylamino)-N-
(7-(hydroxyamino)-7-oxoheptyl)pyrimidine-5-carboxamide |
|
R10793 |
(-)-JQ1 |
The bromodomain and extra terminal domain (BET) family of proteins, including BR
|
R10794 |
Capadenoson; BAY 68-4986 |
Capadenoson (BAY 68-4986) is a new adenosine A1 receptor agonist.
|
R10797 |
CWHM-12 |
CWHM-12是αV整联蛋白的有效抑制剂,抑制αvβ8,αvβ3,αvβ6和αvβ1的 IC50 值分别为0.2,0.8,1.5,1.8 nM。
|
R10799 |
LCL161 Enantiomer |
LCL161 is an orally bioavailable second mitochondrial-derived activator of caspa
|
R10801 |
Deltarasin |
Deltarasin is a small molecular inhibitor of KRAS-PDEδ interaction with Kd of 38
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