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目录号 | 产品名称 | 产品描述 |
R10552 | Fludarabine phosphate | Fludarabine Phosphate is an analogue of adenosine and deoxyadenosine, which is a |
R10553 | Venetoclax; ABT199 | Venetoclax (ABT-199; GDC-0199) 是一种高效,有选择性和口服活性的 Bcl-2 抑制剂,Ki 小于0.01 nM。 |
R10554 | Ipatasertib;GDC-0068; RG7440 | Ipatasertib (GDC-0068) 是一种选择性,竞争性的 pan-Akt 抑制剂,抑制 Akt1,Akt2,Akt3 的 IC50 分别为 5,18 |
R10555 | PF-06687859; RG-3039 | RG3039 (PF-06687859) 是具有口服活性,可渗透大脑的 DcpS 抑制剂, IC50 值为 0.069 nM。 |
R10556 | LY2835219 Intermediate 1 | LY2835219 is a potent and selective inhibitor of CDK4 and CDK6 with IC50 of 2 nM |
R10557 | Fruquintinib; HMPL-013 | Fruquintinib (HMPL-013) 是有效,选择性的 VEGFR 1/2/3 抑制剂,IC50 值分别为33,0.5, |
R10558 | 3R,4S,5S-tert-butyl 3-methoxy-5-methyl-4-; methylaminoheptanoatehydrochloride | |
R10559 | MK-5172 Intermediate 1 | |
R10560 | MK-5172 Intermediate 2 | |
R10561 | ABT199 Intermediate 1 | |
R10562 | TP-353 | 中文名称:TP-353 CAS号:1253799-29-9 中文别名: 英文名称:2-Benzyloxy-3-dibenzylamino-5-fluoro-6- |
R10563 | LHW090-A7 | LHW090-A7 is a compound developed as an inhibitor of neutral endopeptidase (NEP) |
R10565 | INCB8761 Intermediate | |
R10568 | Fedratinib; TG101348 | Fedratinib (TG-101348) 是 JAK2 的选择性抑制剂, IC50为3 nM,比对JAK1和JAK3的选择性高35,334倍。 |
R10569 | Pelitinib | Pelitinib (EKB-569) is a potent irreversible EGFR inhibitor with IC50 of 38.5 nM |
R10570 | Safinamide mesylate | Safinamide Mesylate is mesylate salt of Safinamide, selectively and reversibly i |
R10571 | 2,3-cyclopentenopyridine | |
R10572 | Belinostat;PXD101 | Belinostat (PXD101)是一种新型HDAC抑制剂,无细胞试验中IC50为27 nM,对耐Cisplatin的肿瘤具有活性。 |
R10573 | 2,3-Cyclohexeno pyridine | |
R10583 | Tenofovir alafenamide (Synonyms: GS-7340) | Tenofovir alafenamide (GS-7340) 是 Tenofovir 的前体,Tenofovir 是一种 HIV-1 核苷酸逆转录酶抑制剂。& |
R10584 | Tenofovir alafenamide fumarate (Synonyms: GS-7340 (fumarate)) | Tenofovir alafenamide fumarate (GS-7340 fumarate) 是 Tenofovir 的前体,Tenofovir 是一种 |
R10585 | AZD3759 | AZD3759 是一种有效的可渗透中枢神经系统的 EGFR 抑制剂。作用于 EGFRwt,EGFRL858R 和 EGFRexon 19Del,IC50 分别为 |
R10586 | Tiplaxtinin;PAI-039 | Tiplaxtinin(PAI-039) is an orally efficacious and selective plasminogen activato |
R10587 | UNC0064-12 | |
R10590 | Kartogenin | Kartogenin is an activator of the smad4/smad5 pathway, and promotes the selectiv |