R10522 |
Blonanserin,AD5423 |
Blonanserin is a relatively selective serotonin (5-HT)2A and dopamine D2 antagon
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R10523 |
Aripiprazole |
Aripiprazole is a novel atypical antipsychotic drug that is reported to be a hig
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R10524 |
Blonanserin Intermediate |
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R10526 |
Anagrelide hydrochloride; BL4162A |
Anagrelide is a drug used for the treatment of essential thrombocytosis.
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R10527 |
Anagrelide Intermediate |
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R10529 |
哌立福新;Perifosine(KRX-0401; NSC 639966; D21266) |
Perifosine是一种有口服活性的 Akt 抑制剂,抑制不同肿瘤细胞系增殖的 IC50 值为0.6-8.9 μM。
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R10531 |
Doripenem (S4661) |
Doripenem是β-内酰胺广谱抗生素,对革兰氏阳性菌、阴性菌和厌氧菌均有效。
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R10532 |
Tebipenem pivoxil; L-084 |
Tebipenem Pivoxil是新型口服碳青霉烯类抗生素。
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R10533 |
Agomelatine (S-20098) |
Agomelatine (S-20098) 是一种 MT1 和 MT2 受体的特异性激动剂,对 CHO-hMT1,HEK-hMT1,CHO-hMT2,HEK-h
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R10534 |
Fosaprepitant dimeglumine (Synonyms: MK-0517; L785298) |
Fosaprepitant dimeglumine(MK-0517)是神经激肽-1受体拮抗剂,可作用于化疗引起的恶心呕吐
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R10535 |
Afatinib dimaleate; BIBW2992 dimaleate |
Afatinib dimaleate (BIBW 2992MA2) 是不可逆的 EGFR 家族抑制剂,抑制EGFRwt,EGFRL858R,EGFRL858R/
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R10536 |
Tofacitinib citrate (Tasocitinib citrate; CP-690550 citrate) |
Tofacitinib citrate是 JAK3/2/1 抑制剂,IC50 分别为1,20 和 112 nM。
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R10537 |
Tasocitinib Intermediate |
Tofacitinib (CP-690550) Citrate is a novel inhibitor of JAK3 with IC50 of 1 nM i
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R10538 |
Carteolol hydrochloride (OPC-1085 hydrochloride) |
Carteolol hydrochloride (OPC-1085 hydrochloride) 是非选择性β肾上腺素受体阻断剂。
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R10539 |
Carteolol Intermediate |
Carteolol HCl is a β-adrenoceptor antagonist, used for the treatment of glaucoma
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R10540 |
Regorafenib monohydrate |
Regorafenib monohydrate 是一种多靶点抑制剂,对VEGFR1/2/3,PDGFRβ,Kit,RET 和 Raf-1 的 IC50 分别为
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R10541 |
Regorafenib Intermediate |
Regorafenib is a multi-target inhibitor for VEGFR1, VEGFR2, VEGFR3, PDGFR??, Kit
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R10542 |
Zearalenone (Synonyms: Mycotoxin F2; Toxin F2) |
Zearalenone 是一种真菌毒素,主要有食物和饲料中的Fusarium产生。在猪、牛、羊体内具有雌激素活性,急性毒性低。会引起幼龄母猪乳房发育早熟或其它雌
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R10543 |
Plerixafor; AMD310 |
Plerixafor (AMD3100) is a chemokine receptor antagonist for CXCR4 and CXCL12-med
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R10544 |
Rabeprazole sodium |
Rabeprazole sodium(LY307640 sodium) is an antiulcer drug in the class of proton
|
R10545 |
CANGRELOR |
Regorafenib is a multi-target inhibitor for VEGFR1, VEGFR2, VEGFR3, PDGFR, Kit,
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R10547 |
Deferasirox |
Deferasirox is a rationally-designed oral iron chelator.
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R10549 |
Azilsartan medoxomil; TAK491 |
Azilsartan Medoxomil is a potent angiotensin II type 1 (AT1) receptor antagonist
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R10550 |
Vorinostat |
Vorinostat (suberoylanilide hydroxamic acid, SAHA) is an HDAC inhibitor with IC5
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R10551 |
Escitalopram oxalate |
Escitalopram Oxalate is a selective serotonin (5-HT) reuptake inhibitor (SSRI) w
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