| R2101037 |
GW779439X |
GW779439X is an inhibitor of cyclin dependent kinase.
|
| R2101038 |
RO2959 hydrochloride |
RO2959 hydrochloride 是一种有效的选择性 CRAC 通道抑制剂,IC50 为 402 nM。RO2959 hydrochloride 是由
|
| R2101039 |
Flupenthixol dihydrochloride |
cis-(Z)-Flupentixol dihydrochloride 是有效、选择性的多巴胺DA D1/D2 受体的拮抗剂,其对D2 受体和 5-HT2A 的
|
| R2101040 |
4BP-TQS |
4BP-TQS is an allosteric agonist of α7 subunit-containing neuronal nicotinic ace
|
| R2101041 |
B355252 |
B355252 is a neuroprotective agent that potentiates nerve growth factor (NGF)-in
|
| R2101042 |
GSK 2830371 |
GSK 2830371 是一种选择性的Wip1磷酸酶 (Wip1 phosphatase)抑制剂,IC50 为 6 nM。
|
| R2101043 |
MONNA |
MONNA is a potent TMEM16A (Anoctamin-1) blocker (IC50 = 80 nM). Exhibits >100
|
| R2101044 |
TAE-1 |
TAE-1 is an inhibitor of amyloid-β fibril formation and aggregation, suggesting
|
| R2101045 |
ML191 |
ML-191 is a potent, selective GPR55 antagonist with 160 nM potency for GPR55 and
|
| R2101046 |
ML336 |
ML-336 is an inhibitor of of the Venezuelan equine encephalitis virus (VEEV) str
|
| R2101047 |
GW280264X |
GW280264X is an ADAM17 inhibitor.
|
| R2101048 |
TM5007 |
TM5007 is a poent inhibitor plasminogen activator inhibitor-1 (PAI-1) with IC50
|
| R2101049 |
CYM2503 |
CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that poten
|
| R2101050 |
YM26734 |
YM-26734 is a rabbit platelet sPLA2 inhibitor that has been used to ameliorate l
|
| R2101051 |
G244-LM |
G244-LM is a potent and specific tankyrase 1/2 inhibitor that inhibits Wnt signa
|
| R2101052 |
VK-II-86 |
VK-II-86 is a selective ryanodine receptor type 2 (RyR2) antagonist.
|
| R2101053 |
ML298 |
ML298 (CID53393915) is a potent, specific inhibitor of Phospholipase D2 (PLD2) w
|
| R2101054 |
SW155246 |
SW155246 is a potent and selective DNMT1 (DNA methyltransferase 1) inhibitor wit
|
| R2101055 |
ML-299 |
ML299 (VU0463568) is a dual inhibitor of PLD1 and PLD2 with IC50 of 6 nM and 20
|
| R2101056 |
VUF11418 |
VUF11418 is a nonpeptidomimetic agonist of the G protein-coupled chemokine recep
|
| R2101057 |
CGS-15943 |
CGS15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor
|
| R2101058 |
NSC177223 |
API-1 (NSC 177223) is a potent inhibitor of Akt that induces GSK3-dependent, β-T
|
| R2101059 |
ML162 |
一种小分子探针,选择性杀死诱导表达突变RAS的细胞;抑制BJeLR(表达HRAS G12V)细胞系,IC50为25 nM,显示出比BJeH LT(不含HRAS
|
| R2101060 |
GSK-843 |
GSK-843 是一种受体相互作用蛋白激酶 3 (RIP3 or RIPK3) 抑制剂,高亲和力结合 RIP3 激酶结构域,IC50 值为 8.6 nM,并抑制
|
| R2101061 |
Imidazenil |
Imidazenil is a GABA-A modulator that blocks the sedative effects without loweri
|