| R2101012 |
Dafadine-A |
Dafadine-A是dafadine类似物,是C. elegans DAF-9 细胞色素P450抑制剂,还能抑制哺乳动物的CYP27A1。
|
| R2101013 |
Fluxapyroxad |
Fluxapyroxad is a broad-spectrum fungicide that inhibits the succinate dehydroge
|
| R2101014 |
WIKI4 |
WIKI4是Wnt/_beta_-catenin信号转到抑制剂,EC50值约75nM。
|
| R2101015 |
PCNA-I 1 |
PCNA-I1 is a proliferating cell nuclear antigen (PCNA) inhibitor. It inhibits gr
|
| R2101016 |
CYM50308 |
CYM50308 是一种有效的,选择性和高亲和力的鞘氨醇-1-磷酸受体 4 (S1P4-R) 激动剂,EC50 为 56 nM。CYM50308 对 S1P4-
|
| R2101017 |
BC-1215 |
BC-1215 是 F-box protein 3 (FBXO3) 的抑制剂,IL-1β 释放时,IC50 值为 0.9 μg/mL。 BC-1215 降低 F
|
| R2101018 |
BC-1258 |
密度 1.2±0.1 g/cm3
沸点 599.9±60.0 °C at 760 mmHg
闪点 316.6±32.9 °C
蒸汽压 0.0±1.7 mmHg
|
| R2101019 |
BMS-191011 |
BMS-191011 (BMS-A) 是一种大电导钙激活钾通道 (large-conductance, Ca2++-activated potassium (m
|
| R2101020 |
CRT0066101 dihydrochloride |
CRT0066101 is a specific inhibitor of all Protein kinase D (PKD) isoforms.
|
| R2101021 |
AA92593 |
AA92593 (Opn4 Antagonist) is a potent antagonist of melanopsin-mediated phototra
|
| R2101022 |
ML335 |
ML335 (CYM 51010, CID-23723457) is an agonist for OPRM1(μ-opioid receptor)-OPRD1
|
| R2101023 |
VK-II-36 |
VK-II-36 is a carvedilol analog that suppresses sarcoplasmic reticulum (SR) Ca(2
|
| R2101024 |
YMU1 |
ML335 (CYM 51010, CID-23723457) is an agonist for OPRM1(μ-opioid receptor)-OPRD1
|
| R2101025 |
ML254 |
ML254 is shown to competitively interact with the MPEP allosteric binding site.
|
| R2101026 |
PU-H54 |
A potent, selective Grp94 inhibitor.
|
| R2101027 |
ML303 |
ML303 是一种吡唑并吡啶类化合物, 是流感病毒非结构蛋白 1 (NS1) 的拮抗剂 (IC90 为 155 nM),其对流感病毒H1N1亚型的 EC50 值
|
| R2101028 |
Nisoxetine hydrochloride |
Nisoxetine hydrochloride 是一种有效的和选择性的去甲肾上腺素转运蛋白 (NET) 的抑制剂,Kd 值为 0.76 nM。Nisoxeti
|
| R2101029 |
ASN03576800 |
ASN03576800 is an inhibitor of the VP40 matrix protein.
|
| R2101030 |
HA-155 |
HA155 (Autotaxin Inhibitor IV), a boronic acid-based compound, inhibits autotaxi
|
| R2101031 |
CYM5520 |
noncompetitive allosteric agonist of S1P2
|
| R2101032 |
CRT5 |
CRT5 (CRT0066051), a pyrazine benzamide, is a potent and selective PKD inhibitor
|
| R2101033 |
BMS453 |
BMS453 (BMS-189453) 是一种合成类维生素 A,是一种 RARβ 激动剂和 RARα/RARγ 拮抗剂。BMS453 主要通过诱导活性 TGFβ
|
| R2101034 |
Mps1-IN-3 |
Mps1-IN-3 是一种有效的,选择性的 MPS1 抑制剂,IC50 值为 50 nM。
|
| R2101035 |
OS-3-106 |
OS-3-106 is a novel dopamine D3 receptor-selective partial agonist.
|
| R2101036 |
NSC-703786 |
A potent, selective antitumour agent through activation the aryl hydrocarbon rec
|