R10555 |
PF-06687859; RG-3039 |
RG3039 (PF-06687859) 是具有口服活性,可渗透大脑的 DcpS 抑制剂, IC50 值为 0.069 nM。
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R10586 |
Tiplaxtinin;PAI-039 |
Tiplaxtinin(PAI-039) is an orally efficacious and selective plasminogen activato
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R10594 |
CID2011756 |
CID-2011756 is a cell-active ATP competitive and specific PKD1 inhibitor that in
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R10600 |
Ampalex; CX-516 |
Ampalex (Ampakine CX516; CX516; BDP 12) is an ampakine and nootropic that acts a
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R10611 |
PD169316 |
PD 169316 是一种高效,细胞透过的,有选择性的 p38 MAP kinase 抑制剂,IC50 值为 89 nM。PD169316 选择性地抑制磷酸化
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R10612 |
RKI-1313 |
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R10613 |
1246535-95-4 |
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R10614 |
HPGDS inhibitor 1 |
HPGDS inhibitor 1 is a novel and selective Hematopoietic Prostaglandin D Synthas
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R10619 |
AT-56 |
AT-56 is am orally active inhibitor of lipocalin-type prostaglandin D synthase (
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R10620 |
ML161 |
ML-161 is an allosteric inhibitor of PAR1 with IC50 of 0.26 μM.
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R10623 |
Etofenamate |
Etofenamate is an anti-inflammatory, anti-arrhythmic amino acid.
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R10625 |
NSI-189 |
NSI-189 is a nootropic and neurogenic research chemical derived from nicotinamid
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R10627 |
ICILIN |
Icilin is a cooling agent that activates the novel cold receptors TRPM8 (CMR1) a
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R10630 |
Siramesine Hydrochloride |
Siramesine Hydrochloride is a selective sigma-2 receptor agonist, which has been
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R10631 |
SiramesineLu-28-179 |
Anti-cancer agent siramesine is a lysosomotropic detergent that induces cytoprot
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R10634 |
Betrixaban |
Betrixaban 是一种口服有效的选择性 factor Xa (fXa) 抑制剂,IC50 为 1.5 nM。
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R10637 |
Methylisoindigotin |
Meisoindigo, a derivative of Indigo naturalis, is a promising agent with in vitr
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R10643 |
VGX-1027 |
VGX-1027 is an orally active immunomodulator. Phase 1.
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R10644 |
Y320 |
Y-320是免疫调节剂,能抑制IL-15刺激CD4 T细胞后的IL-17生成,IC50为20到60 nM。
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R10645 |
Atglistatin |
Atglistatin 是一种选择性的脂肪甘油三酯脂酶 (ATGL) 抑制剂,体外抑制脂解作用,IC50 为 0.7 μM。
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R10646 |
Ametantrone ;NSC196473 |
Ametantrone (AM) is a synthetic 9,10-anthracenedione bearing two (hydroxyethylam
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R10649 |
P7C3 |
P7C3 is a potent proneurogenic and neuroprotective chemical that targets NAMPT e
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R10656 |
CP-640186;CP640186 |
CP-640186 是一种有效且可透过细胞的 乙酰辅酶A羧化酶 (ACC) 抑制剂,抑制大鼠肝脏 ACC1 和大鼠骨骼肌 ACC2 的 IC50为 53 nM
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R10657 |
CID797718 |
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R10662 |
TTP22 |
TTP 22 is a high affinity, casein kinase 2 (CK2) inhibitor (IC50= 0.1uM, Ki= 40n
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