| R2030279 |
PND-1186 (VS-4718; SR-2516) |
PND-1186 (VS-4718; SR-2516) 是有效可逆的 FAK 抑制剂,细胞试验中的 IC50 为1.5 nM。
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| R2030280 |
SB742457;Intepirdine (SB-742457; GSK-742457; RVT-101) |
Intepirdine (SB742457) 是5-HT6受体拮抗剂,pKi为9.63,比对其它受体的抑制性高100倍以上。
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| R2030281 |
TGX-221 |
TGX-221 是一种高效的、选择性的、细胞膜渗透的 PI3K p110β 抑制剂,常用于癌症治疗。
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| R2030282 |
VR23 |
VR23有效抑制胰蛋白酶样蛋白酶 (IC50=1nM), 胰凝乳蛋白酶样蛋白酶 (IC50 =50-100 nM), 和caspase样蛋白酶 (IC50 =3
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| R2030283 |
OTX008 (Calixarene 0118; PTX008) |
OTX008 是一个半乳糖凝集素 1 (galectin-1) 的选择性抑制剂。
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| R2030284 |
1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-methylsulfanyl-2-prop-2-enylpyrazolo[3,4-d]pyrimidin-3-one |
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| R2030285 |
4-bromopyridazine,hydrobromide |
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| R2030286 |
ethyl 4'-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2,3,4,5-tetrahydro-[1,1'-biphenyl]-4-carboxylate |
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| R2030292 |
(3-chloropyrazin-2-yl)methanamine hydrochloride |
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| R2030293 |
4-Chlorothieno[3,2-d]pyrimidine |
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| R2030294 |
7-BROMO-4-CHLOROTHIENO[3,2-D]PYRIMIDINE |
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| R2030295 |
6-bromo-4-chlorothieno[3,2-d]pyrimidine |
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| R2030296 |
4-BENZYLOXYBUTYRIC ACID |
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| R2030297 |
2-Pyridineacetic acid, 6-methyl- (9CI) |
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| R2030298 |
4-amino-2-chloronicotinaldehyde |
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| R2030299 |
3-IODO-4-METHOXY-PYRIDIN-2-YLAMINE |
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| R2030300 |
2-AMino-3-forMyl-4-chloropyridine |
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| R2030301 |
1-(4-BROMOPHENYL)PIPERAZINE |
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| R2030302 |
tert-butyl 4-(4-bromophenyl)piperazine-1-carboxylate |
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| R2030303 |
5-Chloro-2-(chloromethyl)pyridine |
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| R2030304 |
(5-chloropyridin-2-yl)methanamine,dihydrochloride |
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| R2030305 |
1-(Aminomethyl)cyclopropanecarboxylic acid hydrochloride |
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| R2030306 |
2-Amino-4-methoxypyridine |
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| R2030307 |
6-Bromo-2-methylpyridin-3-ol |
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| R2030308 |
6-Chloropyridazine-3-carboxylic acid |
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