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目录号 产品名称 产品描述
R10311 E7080; E7080; Lenvatinib Intermediate3 Neratinib (HKI-272) is a highly selective HER2 and EGFR inhibitor with IC50 of 5
R10312 E7080; E7080; Lenvatinib Intermediate4 Neratinib (HKI-272) is a highly selective HER2 and EGFR inhibitor with IC50 of 5
R10313 KU0059436; AZD2281; OlaparibIntermediate Olaparib (AZD2281, KU0059436) is a selective inhibitor of PARP1/2 with IC50 of 5
R10314 PD0332991; PD0332991; Palbociclib Palbociclib (PD0332991) Isethionate is a highly selective inhibitor of CDK4/6 wi
R10315 PD0332991; Palbociclib Intermediate1 Palbociclib (PD0332991) Isethionate is a highly selective inhibitor of CDK4/6 wi
R10316 PD0332991; Palbociclib Intermediate2 Palbociclib (PD0332991) Isethionate is a highly selective inhibitor of CDK4/6 wi
R10317 PD0332991; Palbociclib Intermediate3 Palbociclib (PD0332991) Isethionate is a highly selective inhibitor of CDK4/6 wi
R10318 Valsartan/sacubitril; LCZ696 Intermediate1 LCZ696, consisting of valsartan and sacubitril in 1:1 molar ratio, is an orally
R10319 Valsartan/sacubitril; LCZ696 Intermediate2 LCZ696, consisting of valsartan and sacubitril in 1:1 molar ratio, is an orally
R10320 Valsartan/sacubitril; LCZ696 Intermediate3 LCZ696, consisting of valsartan and sacubitril in 1:1 molar ratio, is an orally
R10321 MS37452
R10322 Ryuvidine Ryuvidine 是一种含有的 SET 结构域的蛋白质 8 (SETD8) 的有效抑制剂,其 IC50 为 0.5 µM,并在体外抑制 H4K20 的甲基化。
R10323 ML190; Indomethacin morpholinylamide
R10329 Elafibranor;GFT505;GFT-505;GFT 505 Elafibranor is an agonist of the peroxisome proliferator-activated receptor-α an
R10330 GFT505; elafibranor E Elafibranor是 PPARα/δ 的激动剂,EC50 分别为 45 和 175 nM。 
R10331 Cabozantinib S-malate (XL184 S-malate; BMS-907351 S-malate) Cabozantinib S-malate (XL184 S-malate) 是一种有效的多受体酪氨酸激酶抑制剂, 抑制VEGFR2,c-Met,Kit,Axl
R10332 Molibresib (Synonyms: GSK 525762A; I-BET 762) Molibresib (GSK 525762A; I-BET 762) 是 BET 溴结构域 抑制剂,IC50 为32.5-42.5 nM。
R10333 Navitoclax (Synonyms: ABT-263) Navitoclax (ABT-263) 是有效,可口服的 Bcl-2 抑制剂,可与Bcl-xL,Bcl-2, Bcl-w等多种Bcl-2家族蛋白结合,Ki 值
R10334 SU6656 SU 6656 is a selective Src family kinase inhibitor with IC50 of 280 nM, 20 nM, 1
R10336 Felbamate; Felbatol Felbamate (Felbatol) is an anticonvulsant drug used in the treatment of epilepsy
R10339 PLX-3397; Pexidartinib Pexidartinib (PLX3397) is an oral, potent mutil-targeted receptor tyrosine kinas
R10341 BS-181 hydrochloride BS-181盐酸盐是CDK7高效选择性抑制剂,IC50值21nM,对CDK1/92/4/5/6/9作用弱。 
R10342 GW 627368 GW627368 (GW627368X) 是前列腺素受体 EP4 高效选择竞争性抑制剂,还对血栓素受体 TP 有亲和力。
R10343 Bikinin; Abrasin Bikinin 是一种非甾体类的,植物性 GSK-3/Shaggy-like kinases 的 ATP 竞争性抑制剂,可激活 BR 信号通路。 
R10344 GW9662 GW9662 is a selective PPAR antagonist for PPARγ with IC50 of 3.3 nM in a cell-fr
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